CHR-6494 TFA
Cat. No.:YN290948
| 产品名称: | CHR-6494 TFA |
| CAS No.: | 1458630-17-5 |
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| 分子量: | 406.362 |
| 分子式: | C18H17F3N6O2 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | CHR-6494 TFA 是一种有效的选择性haspin抑制剂,IC50值为 2 nM。CHR-6494 TFA 能够抑制组蛋白 H3T3 的磷酸化。CHR-6494 TFA 诱导黑色素瘤、乳腺癌等肿瘤细胞凋亡 (apoptosis)。CHR-6494 TFA 可用于癌症的研究。 |
| IC50和靶点: | [{name:"haspin:2 nM (IC50)"}] |
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