Zatebradine
Cat. No.:YN360424
| 产品名称: | Zatebradine |
| CAS No.: | 85175-67-3 |
| Chemical Name: | |
| Synonyms: | UL-FS-49 free base; UL-FS-49CL free base |
| 分子量: | 456.57 |
| 分子式: | C₂₆H₃₆N₂O₅ |
| SMILES: | O=C1N(CCCN(CCC2=CC=C(OC)C(OC)=C2)C)CCC3=CC(OC)=C(OC)C=C3C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Zatebradine (UL-FS-49 (free base); UL-FS-49CL (free base)) 是一种高效的HCN Channel抑制剂,其IC50值为 1.96 µM。Zatebradine 会阻止通过人类HCN1,HCN2,HCN3和HCN4通道的缓慢内向电流,其IC50值分别为 1.83 µM,2.21 µM,1.90 µM 和 1.88 µM。_x000D_ . |
| IC50和靶点: | |
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| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |