Mepazine hydrochloride
Cat. No.:YN370919
| 产品名称: | Mepazine hydrochloride |
| CAS No.: | 2975-36-2 |
| Chemical Name: | |
| Synonyms: | Pecazine hydrochloride |
| 分子量: | 346.92 |
| 分子式: | C₁₉H₂₃ClN₂S |
| SMILES: | CN1CC(CN2C3=C(C=CC=C3)SC4=CC=CC=C24)CCC1.[H]Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Mepazine hydrochloride (Pecazine hydrochloride) 是一种有效的选择性MALT1蛋白酶抑制剂。Mepazine hydrochloride 抑制全长 GSTMALT1 和 GSTMALT1 325-760 段的IC50分别为 0.83 和 0.42 μM。Mepazine hydrochloride 通过增强细胞凋亡 (apoptosis) 来影响 ABC-DLBCL 细胞的生存能力。 |
| IC50和靶点: | |
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