Ropinirole
Cat. No.:YN1730162
| 产品名称: | Ropinirole |
| CAS No.: | 91374-21-9 |
| Chemical Name: | |
| Synonyms: | 罗匹尼罗; SKF 101468 |
| 分子量: | 260.37 |
| 分子式: | C16H24N2O |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Ropinirole (SKF 101468) 是一种口服有效的D3/D2受体激动剂,对 D2受体的Ki为 29 nM。Ropinirole 对 hD2,hD3和 hD4受体的pEC50分别为 7.4、8.4 和 6.8。Ropinirole 对 D1受体没有亲和力。Ropinirole 具有用于帕金森氏病潜力。 |
| IC50和靶点: | [{name:"D2 Receptor:29 nM (Ki)"},{name: "hD2 Receptor:7.4 (pEC50)"},{name: "hD3 Receptor:8.4 (pEC50)"},{name: "hD4.4 Receptor:6.8 (pEC50)"}] |
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| Clinical Trial: | |
| Solvent & Solubility: |