ULK-101
Cat. No.:YN280028
| 产品名称: | ULK-101 |
| CAS No.: | 2443816-45-1 |
| Chemical Name: | |
| Synonyms: | ULK-101; ULK 101; ULK101 |
| 分子量: | 460.45 |
| 分子式: | C₂₂H₁₆F₄N₄OS |
| SMILES: | FC1=CC=C(C(C=N2)=CN3C2=C(C4=CSC(C(N[C@@H](C5CC5)C(F)(F)F)=O)=C4)C=N3)C=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | ULK-101 是一个有效的、选择性的ULK1抑制剂,其在体外测得的对 ULK1和 ULK2 的IC50值分别为 1.6 nM 和 30 nM。ULK-101 抑制自噬,使癌细胞对营养胁迫敏感。 |
| IC50和靶点: | [{name:"ULK1:1.6 nM (IC50)"},{name: "ULK2:30 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |