BMS-345541
Cat. No.:YN410011
| 产品名称: | BMS-345541 |
| CAS No.: | 445430-58-0 |
| Chemical Name: | |
| Synonyms: | BMS345541,IKK Inhibitor III,BMS-345541 free base |
| 分子量: | 255.32 |
| 分子式: | C₁₄H₁₇N₅ |
| SMILES: | CC1=CN=C2C(NCCN)=NC3=CC=C(C)C=C3N21 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | BMS-345541 是一种选择性的IKK催化亚基 IKK-1 和 IKK-2 抑制剂,抑制IKK-2和IKK-1,IC50值分别为 0.3 μM 和 4 μM。BMS-345541 与 IKK 的变构位点结合。 |
| IC50和靶点: | [{name:"IKK-2:0.3 μM (IC50)"},{name: "IKK-1:4 μM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |