HPN-01
Cat. No.:YN410183
| 产品名称: | HPN-01 |
| CAS No.: | 928655-63-4 |
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| 分子量: | 401.87 |
| 分子式: | C19H16ClN3O3S |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | HPN-01 是一种有效选择性的IKK抑制剂,对 IKK-α、IKK-β 和 IKK-ε 的pIC506.4、7.0 和 <4.8。HPN-01 比 50 多种其他激酶显示出大于50倍的选择性,包括 ALK5、CDK-2、EGFR、ErbB2、GSK3β、PLK1、Src 和 VEGFR-2。 |
| IC50和靶点: | [{name:"IKK-α:6.4 (pIC50)"},{name: "IKK-β:7.0 (pIC50)"},{name: "IKK-ε:<4.8 (pIC50)"}] |
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