INH14
Cat. No.:YN410022
| 产品名称: | INH14 |
| CAS No.: | 200134-22-1 |
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| 分子量: | 240.30 |
| 分子式: | C₁₅H₁₆N₂O |
| SMILES: | O=C(NC1=CC=CC=C1)NC2=CC=C(CC)C=C2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | INH14 是IKKα/IKKβ的抑制剂,IC50值分别为 8.97 和 3.59 μM。INH14 抑制 IKKα/β 依赖性TLR炎症反应。抑制 TAK1/TAB1 的下游和 NF-kB 信号通路。具有抗炎和抗癌作用。 |
| IC50和靶点: | [{name:"IKKβ:3.59 μM (IC50)"},{name: "IKKα:8.97 μM (IC50)"}] |
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