HS014
Cat. No.:YN321874
| 产品名称: | HS014 |
| CAS No.: | 207678-81-7 |
| Chemical Name: | |
| Synonyms: | Ac-CEH-{D-2Nal}-RWGCPPKD-NH2 (Disulfide bridge:Cys1-Cys8) |
| 分子量: | 1563.76 |
| 分子式: | C₇₁H₉₄N₂₀O₁₇S₂ |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | HS014 是一种高效、选择性的黑素皮质素-4(MC4)受体拮抗剂,对人 MC4、MC1、MC3 和 MC5 受体的Ki值分别为 3.16、108、54.4 和 694 nM。HS014 调节吗啡对小鼠行为的影响。HS014 增加自由喂养大鼠的食物摄取量。 |
| IC50和靶点: | |
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| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |