Pimavanserin tartrate
Cat. No.：YN320889
CAS No. ：706782-28-7
| 产品名称: | Pimavanserin tartrate |
| CAS No.: | 706782-28-7 |
| Chemical Name: | N-[(4-Fluorophenyl)methyl]-N-(1-methyl-4-piperidinyl)-N'-[[4-(2-methylpropoxy)phenylurea (2R,3R)-2,3-Dihydroxybutanedioate |
| Synonyms: | ACP-103 tartrate |
| 分子量: | 1005.20 |
| 分子式: | C₅₄H₇₄F₂N₆O₁₀ |
| SMILES: | O=C(NCC1=CC=C(OCC(C)C)C=C1)N(CC2=CC=C(F)C=C2)C3CCN(C)CC3.O=C(O)[C@H](O)[C@@H](O)C(O)=O.O=C(NCC4=CC=C(OCC(C)C)C=C4)N(CC5=CC=C(F)C=C5)C6CCN(C)CC6 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Pimavanserin tartrate (ACP-103) 是一种有效的5-HT 2A受体反向激动剂，pIC50和pKi值分别为8.73和9.3。 |
| IC50和靶点: | [{name:"5-HT2A Receptor:8.73 (pIC50)"},{name: "5-HT2A Receptor:9.3 (pKi)"}] |
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| Solvent & Solubility: |
Doggrell, S.: Drug. Fut., 32, 1007 (2007)
Hacksell, U., et al.: Neuro. Res., No vol. given, 1 (2014)
Newman-Tancredi, A. & Kleven, M.: Psychopharmacology, 216, 451 (2011)
Price, D., et al.: Behav. Pharma., 23, 426 (2012)
