Ecopipam
Cat. No.:YN380323
CAS No. :112108-01-7
产品名称: | Ecopipam |
CAS No.: | 112108-01-7 |
Chemical Name: | |
Synonyms: | SCH 39166 |
分子量: | 313.82 |
分子式: | C19H20ClNO |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Ecopipam (SCH 39166) 是一种有效的、选择性、具有口服活性的多巴胺D1/D5受体拮抗剂,Ki值分别为 1.2 nM 和 2.0 nM。Ecopipam 对 D2、D4、5-HT 和 α2a 受体 (Ki=0.98,5.52,0.08 和 0.73 μM) 显示出超过 40 倍的选择性。Ecopipam 可用于精神分裂症和肥胖症的研究。 |
IC50和靶点: | |
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Clinical Trial: | |
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