MIPS521
Cat. No.：YN322166
CAS No. ：1146188-19-3
| 产品名称: | MIPS521 |
| CAS No.: | 1146188-19-3 |
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| 分子量: | 449.8 |
| 分子式: | C19H10ClF6NOS |
| SMILES: | NC1=C(C(=O)C2=CC=C(Cl)C=C2)C(=CS1)C3=CC(=CC(=C3)C(F)(F)F)C(F)(F)F |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | MIPS521 是腺苷受体 (A1AR) 的正向变构调节剂。MIPS521 还具有较低的 A1AR 变构亲和力 (pKB=4.95; KB=11 μM)。MIPS521 通过调节大鼠脊髓中内源性腺苷水平的升高，在体内表现出减轻疼痛的作用。 |
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