(S)-(+)-Dimethindene maleate
Cat. No.：YN322239
CAS No. ：136152-65-3
| 产品名称: | (S)-(+)-Dimethindene maleate |
| CAS No.: | 136152-65-3 |
| Chemical Name: | N,N-Dimethyl-3-[(1S)-1-(2-pyridinyl)ethyl]-1H-indene-2-ethanamine Maleate; (+)-N,N-Dimethyl-3-[1-(2-pyridinyl)ethyl]-1H-Indene-2-ethanamine-(Z)-2-butenedioate; |
| Synonyms: | |
| 分子量: | 408.49 |
| 分子式: | C24H28N2O4 |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | (S)-(+)-Dimethindene maleate 是一种有效的选择性毒蕈碱M2受体拮抗剂 (pA2= 7.86/7.74;pKi= 7.78)。(S)-(+)-Dimethindene maleate 对毒蕈碱 M1(pA2= 6.83/6.36; pKi= 7.08)，M3(pA2= 6.92/6.96; pKi= 6.70) 和 M4(pKi= 7.00) 受体的亲和力较低。(S)-(+)-Dimethindene maleate 也是一种组胺 H1受体 (histamine H1recep |
| IC50和靶点: | [{name:"mAChR2:7.78 (pKi)"},{name: "mAChR1:7.08 (pKi)"},{name: "mAChR4:7.00 (pKi)"},{name: "mAChR3:6.70 (pKi)"},{name: "H1 Receptor:7.48 (pA2)"}] |
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| Solvent & Solubility: |
