FK888
Cat. No.:YN322244
| 产品名称: | FK888 | 
| CAS No.: | 138449-07-7 | 
| Chemical Name: | |
| Synonyms: | FK-888; FK 888; FK888. | 
| 分子量: | 588.7 | 
| 分子式: | C36H36N4O4 | 
| SMILES: | O=C([C@H]1N(C(C2=CN(C)C3=C2C=CC=C3)=O)C[C@H](O)C1)N[C@@H](CC4=CC=C5C=CC=CC5=C4)C(N(C)CC6=CC=CC=C6)=O | 
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. | 
| 运输: | Room temperature in continental US; may vary elsewhere. | 
| 产品描述: | FK888 是一种有效的、选择性的、高亲和力的二肽NK1受体拮抗剂。FK888 取代 [3H]-SP 结合,Ki值为 0.69 nM 和 0.45 microM。FK888 还在静脉内和口服给药后抑制 SP 诱导的豚鼠气道水肿。 | 
| IC50和靶点: | |
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| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |