Safrazine
Cat. No.:YN380542
产品名称: | Safrazine |
CAS No.: | 2416910-82-0 |
Chemical Name: | |
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分子量: | 324.424 |
分子式: | C20H24N2O2 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | AChE/BChE/MAO-B-IN-1 (Compound 10) 是一种可逆的、非时间依赖的AChE、BChE和MAO-B抑制剂,对 hAChE、hBChE 和 hMAO-B 的IC50分别为 7.31、0.56 和 26.1 μM。AChE/BChE/MAO-B-IN-1 能透过血脑屏障,具有神经保护作用且无细胞毒性。 |
IC50和靶点: | [{name:"MAO-B:26.1 μM (IC50)"},{name: "hAChE:7.31 μM (IC50)"},{name: "hBChE:0.56 μM (IC50)"}] |
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