AZ13705339 hemihydrate
Cat. No.:YN290671
| 产品名称: | AZ13705339 hemihydrate |
| CAS No.: | 2016806-57-6 |
| Chemical Name: | |
| Synonyms: | AZ 13705339 |
| 分子量: | 629.75 |
| 分子式: | C33H36FN7O3S |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | AZ13705339 是一种高效且具有选择性的PAK1抑制剂,对PAK1和 pPAK1 的IC50分别为 0.33 nM 和 59 nM。AZ13705339 对PAK1和PAK2具有结合亲和力,Kd分别为 0.28 nM 和 0.32 nM。AZ13705339 可用于癌症研究。 |
| IC50和靶点: | [{name:"PAK2:0.32 nM (Kd)"},{name: "PAK1:0.28 nM (Kd)"},{name: "PAK1:0.33 nM (IC50)"},{name: "pPAK1:59 nM (IC50)"}] |
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| Clinical Trial: | |
| Solvent & Solubility: |