NFPS
Cat. No.:YN360187
| 产品名称: | NFPS |
| CAS No.: | 405225-21-0 |
| Chemical Name: | |
| Synonyms: | (±)-NFPS |
| 分子量: | 393.45 |
| 分子式: | C₂₄H₂₄FNO₃ |
| SMILES: | OC(CN(C)CCC(C1=CC=C(F)C=C1)OC2=CC=C(C3=CC=CC=C3)C=C2)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | NFPS 是一种选择性,非竞争性甘氨酸转运蛋白-1 (GlyT1) 抑制剂,对 hGlyT1 和 rGlyT1 的IC50分别为 2.8 nM 和 9.8 nM。NFPS 通过 glyR alpha1 亚基在瞬时局灶性脑缺血和再灌注的大鼠模型中发挥神经保护作用。 |
| IC50和靶点: | [{name:"hGlyT1:2.8 nM (IC50)"},{name: "rGlyT1:9.8 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |