TC-MCH 7c
Cat. No.:YN320329
| 产品名称: | TC-MCH 7c |
| CAS No.: | 864756-35-4 |
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| 分子量: | 408.47 |
| 分子式: | C₂₄H₂₅FN₂O₃ |
| SMILES: | O=C1N(C=CC(OCC2=CC=C(F)C=C2)=C1)C3=CC=C(OCCN4CCCC4)C=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | TC-MCH 7c 是一种苯基吡啶酮衍生物,一种口服有效的,选择性的且可穿透血脑屏障的MCH1R拮抗剂,对 hMCH1R 的IC50为 5.6 nM。TC-MCH 7c 对人和小鼠 MCH1R 的Ki分别为 3.4 nM 和 3.0 nM。 |
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