Spinorphin
Cat. No.：YN483825
CAS No. ：137201-62-8
| 产品名称: | Spinorphin |
| CAS No.: | 137201-62-8 |
| Chemical Name: | L-leucyl-L-valyl-L-valyl-L-tyrosyl-L-prolyl-L-tryptophyl-L-threonine |
| Synonyms: | LVV-hemorphin-4 |
| 分子量: | 877.04 |
| 分子式: | C₄₅H₆₄N₈O₁₀ |
| SMILES: | C[C@@H](O)[C@@H](C(O)=O)NC([C@H](CC1=CNC2=CC=CC=C12)NC([C@H]3N(C([C@H](CC4=CC=C(C=C4)O)NC([C@H](C(C)C)NC([C@H](C(C)C)NC([C@H](CC(C)C)N)=O)=O)=O)=O)CCC3)=O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Spinorphin 是脑非肽降解酶的抑制剂。Spinorphin 抑制氨基肽酶、二肽基氨基肽酶III、血管紧张素转换酶和脑非肽酶。Spinorphin 具有镇痛活性。 |
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Yamamoto, Y., Ono, H., Ueda, A., et al.Spinorphin as an endogenous inhibitor of enkephalin-degrading enzymes: Roles in pain and inflammationCurr. Protein Pept. Sci.3(6),587-599(2002)
Honda, M., Okutsu, H., Matsuura, T., et al.Spinorphin, an endogenous inhibitor of enkephalin-degrading enzymes, potentiates leu-enkephalin-induced anti-allodynic and antinociceptive effects in miceJpn. J. Pharmacol.87(4),261-267(2001)
