ELA-21 (human)
Cat. No.:YN484059
产品名称: | ELA-21 (human) |
CAS No.: | 2245073-05-4 |
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分子量: | 2587.14 |
分子式: | C₁₁₂H₁₈₄N₄₀O₂₅S₃ |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | ELA-21 (human) 是一种apelin受体激动剂,pKi为 8.52。ELA-21 (human) 在亚纳摩尔效价下,完全抑制 Forskolin 诱导的 cAMP 产生,并刺激 β-arrestin 募集。ELA-21 (human) 也是 G 蛋白依赖性和非依赖性途径的激动剂。 |
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