BI-0115
Cat. No.:YN1720151
| 产品名称: | BI-0115 |
| CAS No.: | 4929-23-1 |
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| 分子量: | 287.74 |
| 分子式: | C15H14ClN3O |
| SMILES: | 暂无 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | BI-0115 是LOX-1的选择性抑制剂(IC50=5.4 µM),阻止细胞摄取氧化低密度脂蛋白。BI-0115 结合通过形成同二聚体配体结合域的二聚体触发受体抑制。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
Schmidt, G.: U.S. (1968), US 3406168 A