SI-2 hydrochloride
Cat. No.:YN480121
| 产品名称: | SI-2 hydrochloride |
| CAS No.: | 1992052-49-9 |
| Chemical Name: | |
| Synonyms: | EPH 116 hydrochloride |
| 分子量: | 301.77 |
| 分子式: | C₁₅H₁₆ClN₅ |
| SMILES: | CN1C(N/N=C(C)/C2=CC=CC=N2)=NC3=CC=CC=C13.Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | SI-2 hydrochloride (EPH 116 hydrochloride) 是SRC-3 SMI: SRC-3的抑制剂,诱导乳腺癌细胞死亡的IC50值为 3-20 nM。SI-2 hydrochloride (EPH 116 hydrochloride) 具有良好的药代动力学特征和改善的毒性,以及可接受的口服可用性。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |