SGC-GAK-1
Cat. No.：YN480750
CAS No. ：2226517-76-4
规格
价格(RMB)
库存
| 产品名称: | SGC-GAK-1 |
| CAS No.: | 2226517-76-4 |
| Chemical Name: | 6-bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine |
| Synonyms: | GAK inhibitor 1 |
| 分子量: | 389.24 |
| 分子式: | C₁₈H₁₇BrN₂O₃ |
| SMILES: | COC1=C(C(OC)=CC(NC2=CC=NC3=CC=C(C=C23)Br)=C1)OC |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | SGC-GAK-1 是一种有效的选择性细胞周期蛋白 G 相关激酶 (GAK) 抑制剂，Ki为 3.1 nM。SGC-GAK-1 是 GAK 的化学探针。 |
| IC50和靶点: | |
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Asquith, C.R.M., Berger, B.-T., Wan, J., et al.SGC-GAK-1: A chemical probe for cyclin G associated kinase (GAK)J. Med. Chem.62(5),2830-2836(2019)
Saul, S., Pu, S.-Y., Zuercher, W.J., et al.Potent antiviral activity of novel multi-substituted 4-anilinoquin(az)olinesBioorg. Med. Chem. Lett.30(16),127284(2020)
