KRM-III
Cat. No.:YN481309
| 产品名称: | KRM-III |
| CAS No.: | 79220-94-3 |
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| 分子量: | 252.33 |
| 分子式: | C₁₅H₁₂N₂S |
| SMILES: | S=C1NC(C2=CC=CC=C2)=CN1C3=CC=CC=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | KRM-III 是一种有效的具有口服活性的 T 细胞抗原受体 (TCR) 抑制剂。KRM-III 抑制TCR和肉豆蔻酸乙酸酯/佛波霉素/离子霉素诱导的 NFAT 核因子活化和 T 细胞增殖,IC50约为 5 μM。抗炎活性。 |
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