Relenopride hydrochloride
Cat. No.：YN380422
CAS No. ：1221416-42-7
规格
价格(RMB)
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| 产品名称: | Relenopride hydrochloride |
| CAS No.: | 1221416-42-7 |
| Chemical Name: | |
| Synonyms: | YKP10811 hydrochloride |
| 分子量: | 529.43 |
| 分子式: | C24H31Cl2FN4O4 |
| SMILES: | O=C(NCC1CCN(CC[C@H](OC(N)=O)C2=CC=C(F)C=C2)CC1)C3=CC(Cl)=C(N)C=C3OC.[H]Cl |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Relenopride (YKP10811) hydrochloride 是一种特异性和选择性的5-HT4受体激动剂 (Ki=4.96 nM)。与5-HT4相比，Relenopride hydrochloride 对 5-HT2A(Ki=600 nM)和5-HT2B(Ki=31 nM) 受体的亲和力分别低 120 倍和 6 倍。Relenopride hydrochloride 增加胃肠运动。 |
| IC50和靶点: | [{name:"5-HT4 Receptor:4.96 nM (Ki)"},{name: "5-HT2A Receptor:600 nM (Ki)"},{name: "5-HT2B Receptor:31 nM (Ki)"},{name: "5-HT2B Receptor:2.1 μM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
