PI-828
Cat. No.：YN420063
CAS No. ：942289-87-4
规格
价格(RMB)
库存
| 产品名称: | PI-828 |
| CAS No.: | 942289-87-4 |
| Chemical Name: | 8-(4-aminophenyl)-2-(4-morpholinyl)-4H-1-benzopyran-4-one |
| Synonyms: | LY 294002 |
| 分子量: | 322.36 |
| 分子式: | C₁₉H₁₈N₂O₃ |
| SMILES: | O=C1C=C(N2CCOCC2)OC3=C(C4=CC=C(N)C=C4)C=CC=C13 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | PI-828 是一种双重PI3K和casein kinase 2(CK2) 抑制剂，抑制p110α，CK2和CK2α2，IC50分别为 173 nM，149 nM 和 1127 nM。 |
| IC50和靶点: | [{name:"p110α:173 nM (IC50)"},{name: "CK2:149 nM (IC50)"},{name: "CK2α2:1.127 μM (IC50)"}] |
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| Solvent & Solubility: |
Gharbi, S.I., Zvelebil, M.J., Shuttleworth, S.J., et al.Exploring the specificity of the PI3K family inhibitor LY294002Biochem. J.404(1),15-21(2007)
