MK-8033
Cat. No.:YN440259
| 产品名称: | MK-8033 |
| CAS No.: | 1001917-37-8 |
| Chemical Name: | |
| Synonyms: | MK 8033;MK8033 |
| 分子量: | 471.53 |
| 分子式: | C₂₅H₂₁N₅O₃S |
| SMILES: | O=S(NCC1=CC=CC=N1)(CC2=CC=C3C(C(C4=CC(C5=CN(N=C5)C)=CN=C4C=C3)=O)=C2)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | MK-8033 是ATP竞争性c-Met/Ron双重抑制剂,对野生型c-Met的IC50为1 nM,对c-Met N1100Y的IC50为2.0 nM。 |
| IC50和靶点: | [{name:"Ron:7 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |