WIN 55,212-2 Mesylate
Cat. No.：YN320716
CAS No. ：131543-23-2
| 产品名称: | WIN 55,212-2 Mesylate |
| CAS No.: | 131543-23-2 |
| Chemical Name: | [(3R)-2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-methanone, monomethanesulfonate |
| Synonyms: | (R)-(+)-WIN 55212 |
| 分子量: | 522.61 |
| 分子式: | C₂₈H₃₀N₂O₆S |
| SMILES: | O=C(C1=C2C=CC=CC2=CC=C1)C3=C(N4[C@@H](COC5=C4C3=CC=C5)CN6CCOCC6)C.CS(=O)(O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | WIN 55,212-2 Mesylate 是一种有效的cannabinoid receptor激动剂，对人重组 CB1 和 CB2 受体的Ki值分别为 62.3 和 3.3 nM。 |
| IC50和靶点: | |
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| Solvent & Solubility: |
Felder, C.C., Joyce, K.E., Briley, E.M., et al.Comparison of the pharmacology and signal transduction of the human cannabinoid CB1 and CB2 receptorsMol. Pharmacol.48(3),443-450(1995)
Ferraro, L., Tomasini, M.C., Gessa, G.L., et al.The cannabinoid receptor agonist WIN 55,212-2 regulates glutamate transmission in rat cerebral cortex: An in vivo and in vitro studyCereb. Cortex11(8),728-733(2001)
Price, T.J., Patwardhan, A., Akopian, A.N., et al.Cannabinoid receptor-independent actions of the aminoalkylindole WIN 55,212-2 on trigeminal sensory neuronsBr. J. Pharmacol.142(2),257-266(2004)
