Palbociclib-propargyl
Cat. No.:YN430157
| 产品名称: | Palbociclib-propargyl |
| CAS No.: | 2366269-23-8 |
| Chemical Name: | |
| Synonyms: | PROTAC CDK6 ligand 1 |
| 分子量: | 485.58 |
| 分子式: | C₂₇H₃₁N₇O₂ |
| SMILES: | O=C1C(C(C)=O)=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC#C)CC4)C=C3)N=C2N1C5CCCC5 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Palbociclib-propargyl 是一种 PROTAC 靶蛋白CDK6的配体,可通过 PEG linker 与 CRBN 配体结合,组成 PROTAC CP-10。CP-10 可降解 CDK6,DC50值 为 2.1 nM。 |
| IC50和靶点: | |
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| Solvent & Solubility: |