KI-7
Cat. No.:YN1740005
| 产品名称: | KI-7 |
| CAS No.: | 1489263-00-4 |
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| 分子量: | 354.40 |
| 分子式: | C₂₃H₁₈N₂O₂ |
| SMILES: | O=C(NC1=CC=CC=C1)C(C2=CN(CC3=CC=CC=C3)C4=C2C=CC=C4)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | KI-7 是一种A2B腺苷受体阳性变构调节剂。KI-7 增强非选择性 A2B 腺苷受体激动剂 NECA 诱导的 cAMP 积累 (EC50=445.8 nM)。KI-7 还增强了选择性 A2B 腺苷受体激动剂 BAY 60-6583 和 adenosine 诱导的 cAMP 积累,EC50分别为 2390 nM 和 2550 nM。 |
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