A2AR-agonist-1
Cat. No.：YN1730081
CAS No. ：41552-95-8
| 产品名称: | A2AR-agonist-1 |
| CAS No.: | 41552-95-8 |
| Chemical Name: | N-[2-(1H-indol-3-yl)ethyl]-adenosine |
| Synonyms: | N-(2-(1H-Indol-3-yl)ethyl)adenosine |
| 分子量: | 410.43 |
| 分子式: | C₂₀H₂₂N₆O₄ |
| SMILES: | OC[C@@H]1[C@H]([C@H]([C@H](N2C=NC3=C2N=CN=C3NCCC4=CNC5=C4C=CC=C5)O1)O)O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | A2AR-agonist-1是一种有效的 A2AR 和ENT1激动剂, Ki值 分别为 4.39和 3.47。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
Chen, J.-B., Liu, E.M., Chern, T.-R., et al.Design and synthesis of novel dual-action compounds targeting the adenosine A(2A) receptor and adenosine transporter for neuroprotectionChem. Med. Chem.6(8),1390-1400(2011)
Kao, Y.H., Lin, M.S., Chen, C.M., et al.Targeting ENT1 and adenosine tone for the treatment of Huntington's diseaseHum. Mol. Genet.26(3),467-478(2017)
