PSB 0777 ammonium
Cat. No.：YN1710026
CAS No. ：2122196-16-9
| 产品名称: | PSB 0777 ammonium |
| CAS No.: | 2122196-16-9 |
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| 分子量: | 500.55 |
| 分子式: | C₁₈H₂₄N₆O₇S₂ |
| SMILES: | OC[C@@H]1[C@H]([C@H]([C@H](N2C=NC3=C(N=C(SCCC4=CC=C(S(=O)([O-])=O)C=C4)N=C32)N)O1)O)O.[NH4+] |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | PSB 0777 ammonium 是一种有效的选择性腺苷A2A受体激动剂，对大鼠和人 A2A受体的Ki值分别为 44.4 nM，360 nM。PSB 0777 ammonium 对大鼠和人的 A1受体的 Ki值分别 ≥10000 nM，541 nM。PSB 0777 ammonium 显示出较差的大脑渗透性和口服生物利用度。PSB 0777 ammonium 具有用于炎性肠病 (IBS) 研究的潜力。 |
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