GNE-049
Cat. No.:YN310092
| 产品名称: | GNE-049 |
| CAS No.: | 1936421-41-8 |
| Chemical Name: | |
| Synonyms: | GNE049;GNE 049 |
| 分子量: | 510.58 |
| 分子式: | C₂₇H₃₂F₂N₆O₂ |
| SMILES: | CC(N1CCC(N(C2CCOCC2)N=C3N4CCCC5=C4C=C(C(F)F)C(C6=CN(C)N=C6)=C5)=C3C1)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | GNE-049 是一种高效的选择性CBP抑制剂,在 TR-FRET 实验中IC50 sub>为 1.1 nM。GNE-049 还抑制BRET和BRD4(1),IC50分别为 12 nM 和 4200 nM。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |