OXFBD04
Cat. No.:YN310222
| 产品名称: | OXFBD04 |
| CAS No.: | 2231747-03-6 |
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| 分子量: | 296.32 |
| 分子式: | C₁₇H₁₆N₂O₃ |
| SMILES: | OC(C1=CC(O)=CC(C2=C(C)ON=C2C)=C1)C3=CC=CN=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | OXFBD04 是一种有效的选择性BRD4抑制剂,IC50为 166 nM。OXFBD04 是一种有效的 BET 溴结构域配体,对 CREBBP 溴结构域具有额外的适度亲和力。OXFBD04 具有抗癌活性。 |
| IC50和靶点: | [{name:"BRD4:166 nM (IC50)"}] |
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