E-7386
Cat. No.:YN310110
产品名称: | E-7386 |
CAS No.: | 1799824-08-0 |
Chemical Name: | (6S,9aS)-8-[[6-[3-(4-Ethyl-1-piperazinyl)-1-azetidinyl]-2-pyridinyl]methyl]-6-[(2-fluoro-4-hydroxyphenyl)methyl]hexahydro-4,7-dioxo-N-(phenylmethyl)-2-(2-propen-1-yl)-2H-pyrazino[2,1-c][1,2,4]triazine-1(6H)-carboxamide |
Synonyms: | E7386 |
分子量: | 725.85 |
分子式: | C₃₉H₄₈FN₉O₄ |
SMILES: | O=C(N([C@](CN1CC2=NC(N3CC(N4CCN(CC)CC4)C3)=CC=C2)([H])N5[C@@H](CC6=CC=C(O)C=C6F)C1=O)N(CC=C)CC5=O)NCC7=CC=CC=C7 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | E-7386 是一种口服有效的 CBP/β-连环蛋白 (CBP/beta-catenin) 调节剂。 |
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Solvent & Solubility: |
Yusaku, H. et al.: Cancer Res 2017
77(13 Suppl):Abstract nr 5172