CBP-IN-1
Cat. No.:YN310117
CAS No. :2222941-37-7
产品名称: | CBP-IN-1 |
CAS No.: | 2222941-37-7 |
Chemical Name: | (6S)-1-(3,4-difluorophenyl)-6-[5-(3,5-dimethyl-4-isoxazolyl)-1-(trans-4-methoxycyclohexyl)-1H-benzimidazol-2-yl]-2-piperidinone |
Synonyms: | CBP-IN-1, CBP/p300-IN-4 |
分子量: | 534.60 |
分子式: | C₃₀H₃₂F₂N₄O₃ |
SMILES: | O=C1N(C2=CC=C(F)C(F)=C2)[C@H](C3=NC4=CC(C5=C(C)ON=C5C)=CC=C4N3[C@H]6CC[C@H](OC)CC6)CCC1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | CBP-IN-1 是一种高效p300/CBP溴结构域抑制剂。 |
IC50和靶点: | |
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Solvent & Solubility: |
Brooks, N., Raja, M., Young, B.W., et al.CCS1477: A novel small molecule inhibitor of p300/CBP bromodomain for the treatment of acute myeloid leukaemia and multiple myelomaBlood134(Supplement 1),2560(2019)