(R)-BAY1238097
Cat. No.:YN310124
CAS No. :1564269-85-7
产品名称: | (R)-BAY1238097 |
CAS No.: | 1564269-85-7 |
Chemical Name: | |
Synonyms: | |
分子量: | 451.56 |
分子式: | C₂₅H₃₃N₅O₃ |
SMILES: | O=C(N1N=C(C2=CC=C(N3CCN(C)CC3)C=C2)C4=CC(OC)=C(OC)C=C4C[C@H]1C)NC |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | (R)-BAY1238097 是BAY1238097 的低活性 R 型异构体。BAY1238097 是一种有效的、BET与组蛋白 结合的选择性抑制剂,通过下调c-Myc水平及下游转录组,在AML (急性髓性白血病) 和MM (多发性骨髓瘤) 模型中表现出较强的抗增殖活性。 |
IC50和靶点: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |