(+)-JQ1 PA
Cat. No.：YN310135
CAS No. ：2115701-93-2
| 产品名称: | (+)-JQ1 PA |
| CAS No.: | 2115701-93-2 |
| Chemical Name: | (6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-N-2-propyn-1-yl-6H -thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide |
| Synonyms: | (+)-JQ1 PA |
| 分子量: | 437.95 |
| 分子式: | C₂₂H₂₀ClN₅OS |
| SMILES: | O=C(NCC#C)C[C@H]1C2=NN=C(C)N2C3=C(C(C)=C(C)S3)C(C4=CC=C(Cl)C=C4)=N1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | (+)-JQ1 PA 是溴结构域和额外末端结构域(BET)抑制剂JQ1的衍生物，其IC50值为 10.4 nM。 |
| IC50和靶点: | |
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| Clinical Trial: | |
| Solvent & Solubility: |
Tyler, D.S., Vappiani, J., Caneque, T., et al.Click chemistry enables preclinical evaluation of targeted epigenetic therapiesScience356(6345),1397-1401(2017)
