IQ-3
Cat. No.:YN350052
| 产品名称: | IQ-3 |
| CAS No.: | 312538-03-7 |
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 341.32 |
| 分子式: | C₂₀H₁₁N₃O₃ |
| SMILES: | O=C(O/N=C1C2=C(C3=NC4=CC=CC=C4N=C3\1)C=CC=C2)C5=CC=CO5 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | IQ-3 是特异性的c-JNK家族抑制剂,对JNK3 的选择性较好。IQ-3 对 JNK1、JNK2 和 JNK3 的Kd值分别为0.24 μM、0.29 μM 和 0.066 μM。 |
| IC50和靶点: | [{name:"JNK3:0.066 μM (Kd)"},{name: "JNK1:0.24 μM (Kd)"},{name: "JNK2:0.29 μM (Kd)"},{name: "CK1δ:0.56 μM (Kd)"},{name: "PI3Kγ:0.43 μM (Kd)"},{name: "MKNK2:1.2 μM (Kd)"}] |
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