BMS-906024
Cat. No.:YN380113
| 产品名称: | BMS-906024 | 
| CAS No.: | 1401066-79-2 | 
| Chemical Name: | |
| Synonyms: | BMS 906024;BMS906024 | 
| 分子量: | 556.50 | 
| 分子式: | C₂₆H₂₆F₆N₄O₃ | 
| SMILES: | O=C(N[C@@H]1C(N(C)C2=CC=CC=C2C(C3=CC=CC=C3)=N1)=O)[C@H](CCC(F)(F)F)[C@H](CCC(F)(F)F)C(N)=O | 
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. | 
| 运输: | Room temperature in continental US; may vary elsewhere. | 
| 产品描述: | BMS-906024 是一种口服有效,选择性的 γ 分泌酶 (γ-secretase; gamma secretase) 抑制剂。BMS-906024 是有效的,泛Notch受体抑制剂,对 Notch1,-2,-3 和 -4 受体的IC50值分别为 1.6 nM,0.7 nM,3.4 nM 和 2.9 nM。BMS-906024 表现广谱抗肿瘤活性。 | 
| IC50和靶点: | |
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| Clinical Trial: | |
| Solvent & Solubility: |