BJE6-106
Cat. No.:YN310145
CAS No. :1564249-38-2
产品名称: | BJE6-106 |
CAS No.: | 1564249-38-2 |
Chemical Name: | |
Synonyms: | B106 |
分子量: | 381.47 |
分子式: | C₂₆H₂₃NO₂ |
SMILES: | O=CC1=C2C(C=CC(C)(C)O2)=CC(CCN3C4=C(C5=C3C=CC=C5)C=CC=C4)=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | BJE6-106 (B106) 是一种有效的选择性PKCδ抑制剂,IC50值为 0.05 μM,BJE6-106 (B106) 靶向 PKCδ 的选择性是 PKC 同工酶 PKCα 的 1000倍 (IC50=50 μM)。_x000D_ BJE6-106 (B106) 可以诱导 caspase 依耐性细胞凋亡 (apoptosis)。BJE6-106 (B106) 具有肿瘤特异性作用。 |
IC50和靶点: | [{name:"PKCδ:0.05 μM (IC50)"},{name: "PKCα:50 μM (IC50)"}] |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |