GW7647
Cat. No.：YN290297
CAS No. ：265129-71-3
| 产品名称: | GW7647 |
| CAS No.: | 265129-71-3 |
| Chemical Name: | 2-[[4-[2-[[(cyclohexylamino)carbonyl](4-cyclohexylbutyl)amino]ethyl]phenyl]thio]-2-methyl-propanoic acid |
| Synonyms: | 2-[[4-[2-[[环己基氨基)羰基](4-环己基丁基)氨基]乙基]苯基]硫基]-2-甲基丙酸 |
| 分子量: | 502.75 |
| 分子式: | C₂₉H₄₆N₂O₃S |
| SMILES: | CC(C)(SC1=CC=C(CCN(C(NC2CCCCC2)=O)CCCCC3CCCCC3)C=C1)C(O)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | GW7647 是一种有效的PPARα激动剂，对人 PPARα,PPARγ 和 PPARδ 的EC50值分别为 6 nM, 1.1 μM 和 6.2 μM。 |
| IC50和靶点: | [{name:"PPARα:6 nM (EC50, Human PPARα)"},{name: "PPARγ:1.1 μM (EC50, Human PPARγ)"},{name: "PPARδ:6.2 μM (EC50, Human PPARδ)"}] |
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| Solvent & Solubility: |
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Brown, P.J., Stuart, L.W., Hurley, K.P., et al.Identification of a subtype selective human PPARα agonist through parallel-array synthesisBioorg. Med. Chem. Lett.11,1225-1227(2001)
