UNC2541
Cat. No.:YN440217
| 产品名称: | UNC2541 | 
| CAS No.: | 1612782-86-1 | 
| Chemical Name: | |
| Synonyms: | UNC2541; UNC-2541; UNC 2541; | 
| 分子量: | 471.57 | 
| 分子式: | C₂₄H₃₄FN₇O₂ | 
| SMILES: | O=C(C(C(NCCCC[C@@H]1N)=N2)=CN=C2NCCCCCCNC1=O)NCC3=CC=C(F)C=C3 | 
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. | 
| 运输: | Room temperature in continental US; may vary elsewhere. | 
| 产品描述: | UNC2541 是一种有效 Mer 酪氨酸激酶 (MerTK) 特异性抑制剂,与 MerTK ATP 结合口袋结合,IC50值为 4.4 nM,对其选择性远高于 Axl,Tyro3 和 Flt3。UNC2541 抑制磷酸化的 MerTK (pMerTK;EC50,510 nM)。 | 
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |