Afloqualone
Cat. No.：YN360889
| 产品名称: | Afloqualone |
| CAS No.: | 56287-74-2 |
| Chemical Name: | 6-amino-2-(fluoromethyl)-3-(2-methylphenyl)-4(3H)-quinazolinone |
| Synonyms: | 氟喹酮; HQ-495 |
| 分子量: | 283.30 |
| 分子式: | C₁₆H₁₄FN₃O |
| SMILES: | O=C1N(C2=CC=CC=C2C)C(CF)=NC3=C1C=C(N)C=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Afloqualone (HQ-495) 是一种 GABA 能试剂，在GABAα receptor的 β 亚型上具有激动剂活性。Afloqualone 具有抗眩晕和镇静作用，这被认为是由于 LVN 神经元部位 GABA 受体的敏感性增加所致。 |
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| Solvent & Solubility: |
Ochiai, T., and Ishida, R.Pharmacological studies on 6-amino-2-fluoromethyl-3-(O-tolyl)-4(3H)-quinazolinone (afloqualone), a new centrally acting muscle relaxant. (II) Effects on the spinal reflex potential and the rigidityJpn. J. Pharmacol.32(3),427-438(1982)
