1-Azakenpaullone
Cat. No.：YN420280
CAS No. ：676596-65-9
| 产品名称: | 1-Azakenpaullone |
| CAS No.: | 676596-65-9 |
| Chemical Name: | 9-bromo-7,12-dihydro-pyrido[3',2':2,3]azepino[4,5-b]indol-6(5H)-one |
| Synonyms: | 1-Akp |
| 分子量: | 328.16 |
| 分子式: | C₁₅H₁₀BrN₃O |
| SMILES: | O=C(NC1=CC=CN=C12)CC3=C2NC4=C3C=C(Br)C=C4 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | 1-Azakenpaullone (1-Akp) 是具有高度选择性的、ATP 竞争性的糖原合成酶激酶3 β (GSK-3β)的抑制剂，其IC50值为 18 nM。 |
| IC50和靶点: | [{name:"GSK-3β:18 nM (IC50)"},{name: "CDK1/cyclin B:2 μM (IC50)"},{name: "CDK5/p25:4.2 μM (IC50)"}] |
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| Solvent & Solubility: |
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