BRD3731
Cat. No.:YN420127
产品名称: | BRD3731 |
CAS No.: | 2056262-07-6 |
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分子量: | 377.52 |
分子式: | C₂₄H₃₁N₃O |
SMILES: | O=C1C2=C(N=C3C([C@]2(C)C4=CC=CC=C4)=C(CC(C)(C)C)NN3)CC(C)(C)C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | BRD3731 是一种选择性的GSK3β抑制剂,抑制 GSK3β 和 GSK3α 的IC50值分别为 15 nM 和 215 nM。BRD3731 可被用于情绪障碍、创伤后应激障碍 (PTSD) 精神障碍、糖尿病和神经退行性障碍的研究。 |
IC50和靶点: | [{name:"GSK-3β:15 nM (IC50)"},{name: "GSK-3α:215 nM (IC50)"}] |
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