EGFR-IN-5
Cat. No.:YN340072
| 产品名称: | EGFR-IN-5 |
| CAS No.: | 2225887-26-1 |
| Chemical Name: | |
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| 分子量: | 571.69 |
| 分子式: | C₃₁H₃₈FN₉O |
| SMILES: | OCC(CC1)CCN1C2=NC(NC3=CC=C(F)C=C3)=NC(C=N4)=C2C=C4NC5=NC=C(N6CCC(N(C)C)CC6)C=C5 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | EGFR-IN-5是EGFR的抑制剂,对EGFR,EGFRL858R,EGFRL858R/T790M和EGFRL858R/T790M/C797S的IC50分别为10.4,1.1,34,7.2 nM。 |
| IC50和靶点: | [{name:"EGFR:10.4 nM (IC50)"},{name: "EGFRL858R:1.1 nM (IC50)"},{name: "EGFRL858R/T790M:34 nM (IC50)"},{name: "EGFRL858R/T790M/C797S:7.2 nM (IC50)"}] |
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