Bruceantinol
Cat. No.:YN340351
产品名称: | Bruceantinol |
CAS No.: | 53729-52-5 |
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分子量: | 606.61 |
分子式: | C30H38O13 |
SMILES: | 暂无 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | Bruceantinol 是一种从鸦胆子中分离出来的苦味素,可抑制辣椒中的辣椒斑驳病毒。Bruceantinol 是一种STAT3抑制剂,对体内外人结直肠癌 (CRC) 模型都具有抗肿瘤活性。Bruceantinol 抑制STAT3DNA 结合能力 (IC50=2.4 pM),抑制组成型和IL-6诱导的STAT3活化,并抑制 MCL-1、PTTG1、survivin 和 c- Myc 的转录。 |
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