BGB-102
Cat. No.:YN340330
| 产品名称: | BGB-102 |
| CAS No.: | 807640-87-5 |
| Chemical Name: | |
| Synonyms: | JNJ-26483327 |
| 分子量: | 457.36 |
| 分子式: | C22H25BrN4O2 |
| SMILES: | CN1CCCCCOC(C(OC)=C2)=CC3=C2N=CN/C3=N\C4=CC(Br)=CC=C4C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | BGB-102 是多重激酶抑制剂,能够抑制EGFR,HER2和HER4,IC50值分别为 9.6 nM,18 nM 和 40.3 nM。 |
| IC50和靶点: | [{name:"EGFR:9.6 nM (IC50)"},{name: "HER2:18 nM (IC50)"},{name: "HER4:40.3 nM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |