JCN037
Cat. No.:YN340144
| 产品名称: | JCN037 |
| CAS No.: | 2305154-31-6 |
| Chemical Name: | |
| Synonyms: | JGK037 |
| 分子量: | 376.18 |
| 分子式: | C₁₆H₁₁BrFN₃O₂ |
| SMILES: | FC1=C(Br)C=CC=C1NC2=C3C=C(OCCO4)C4=CC3=NC=N2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | JCN037 (JGK037) 是有效的、共价的、能透过血脑屏障的EGFR抑制剂,对 EGFR、p-wtEGFR 和 pEGFRvⅢ 的IC50值分别为 2.49 nM、3.95 nM 和4.48 nM。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |